Affinity DataEC50: 0.0300nMAssay Description:Agonist activity at Ah receptor in genetically engineered mouse cells expressing firefly luciferase gene by CALUX transactivational assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0300nMAssay Description:Agonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 0.0300nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0580nMAssay Description:Activation of AhR in mouse NIH3T3 cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual-lu...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0971nMAssay Description:Agonist activity at EGFP-tagged human AhR transfected in HEK293 cells assessed as induction of nuclear translocation incubated for 45 mins by fluores...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.137nMAssay Description:Agonist activity at human AHR in HEK293 cells assessed as nuclear translocation over cytosol incubated for 45 mins by Hoechst staining based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.161nMAssay Description:Agonist activity at human AHR in HEK293 cells assessed as nuclear translocation over cytosol incubated for 45 mins by Hoechst staining based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.189nMAssay Description:Agonist activity at human AHR in HEK293 cells assessed as nuclear translocation over cytosol incubated for 45 mins by Hoechst staining based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.200nMAssay Description:Activation of human AhR expressed in Saccharomyces cerevisiae YCM3 coexpressing ARNT incubated for 18 hrsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.214nMAssay Description:Agonist activity at EGFP-tagged human AhR transfected in HEK293 cells assessed as induction of nuclear translocation incubated for 45 mins by fluores...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.260nMAssay Description:Agonist activity at AhR in human HepG2 cells assessed as induction of CYP1A1 expression after 24 hrs by ethoxyresorufin-O-deethylase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.270nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.275nMAssay Description:Agonist activity at human AHR in HEK293 cells assessed as nuclear translocation over cytosol incubated for 45 mins by Hoechst staining based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.297nMAssay Description:Agonist activity at human AHR in HEK293 cells assessed as nuclear translocation over cytosol incubated for 45 mins by Hoechst staining based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.304nMAssay Description:Agonist activity at EGFP-tagged human AhR transfected in HEK293 cells assessed as induction of nuclear translocation incubated for 45 mins by fluores...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.340nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.340nMAssay Description:Agonist activity at human AHR in HEK293 cells assessed as nuclear translocation over cytosol incubated for 45 mins by Hoechst staining based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.389nMAssay Description:Agonist activity at EGFP-tagged human AhR transfected in HEK293 cells assessed as induction of nuclear translocation incubated for 45 mins by fluores...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.440nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.447nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 0.468nMAssay Description:Agonist activity at EGFP-tagged human AhR transfected in HEK293 cells assessed as induction of nuclear translocation incubated for 45 mins by fluores...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.511nMAssay Description:Agonist activity at EGFP-tagged human AhR transfected in HEK293 cells assessed as induction of nuclear translocation incubated for 45 mins by fluores...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 0.700nMAssay Description:Activation of AhR in human HaCaT cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual-luc...More data for this Ligand-Target Pair
Affinity DataEC50: 0.830nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.17nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Agonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.48nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at AhR (unknown origin) transfected in human AZ-AHR reporter cells derived from human HepG2 cells incubated for 4 hrs by luciferase ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at AhR in human HepG2 cells assessed as induction of CYP1A1 expression after 24 hrs by ethoxyresorufin-O-deethylase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at AHR in human HepG2 cells incubated for 4.5 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at AHR in human HepG2 cells incubated for 4.5 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Agonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Activation of AhR in human HepG2 cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual-luc...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Concentration of the compound to bind to human AhR-modied electrodeMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Activation of human AhR expressed in Saccharomyces cerevisiae YCM3 coexpressing ARNT incubated for 18 hrsMore data for this Ligand-Target Pair
Affinity DataEC50: 6.61nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 8.40nMAssay Description:Agonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Activation of human AhR expressed in Saccharomyces cerevisiae YCM3 coexpressing ARNT incubated for 18 hrsMore data for this Ligand-Target Pair
Affinity DataEC50: 9.60nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at AhR in mouse Hepa2Dluc cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 11.5nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 15.1nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 15.5nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 17.0nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair